Biological and Pharmaceutical Bulletin · 2010 · in vitro
On excised hairless-mouse skin, glyceryl monocaprylate combined with isopropyl myristate synergistically enhanced pentazocine permeation; permeability rose with glyceryl monocaprylate up to 10% w/w, and X-ray diffraction showed disappearance of the long lamellar order of stratum corneum lipids, indicating barrier-lipid disruption.







